| Compound / class | WADA category | Notes |
|---|---|---|
| Somatropin (GH) | S2 — Peptide hormones | Prohibited at all times |
| GH-releasing factors: sermorelin, tesamorelin, CJC-1295 variants | S2 — Peptide hormones | Releasing factors prohibited at all times |
| GHRP family: ipamorelin, GHRP-2, GHRP-6, hexarelin | S2 — Peptide hormones | Ghrelin receptor agonists prohibited |
| Ibutamoren (MK-677) | S2 — Peptide hormones | GH secretagogue, prohibited |
| IGF-1 and analogs: LR3, DES, MGF, PEG-MGF | S2 — Peptide hormones | Growth factors prohibited |
| Erythropoietin (EPO) | S2 — Peptide hormones | ESAs prohibited at all times |
| HCG and HMG | S2 — Peptide hormones | Prohibited at all times in males |
| Gonadorelin, triptorelin | S2 — Peptide hormones | GnRH-related releasing factors |
| Insulin | S2 — Peptide hormones | Prohibited except with therapeutic use exemption |
| AICAR | S4 — Hormone and metabolic modulators | AMPK activator, prohibited |
| Synthetic oxygen carriers and any non-approved substance | Section 0 / S0 categories | Any drug not approved for human therapeutic use is prohibited by default |
This table is a navigation aid into the entry pages, which carry full evidence and safety context for each compound.
Evidence tier: Approved medicine · Last reviewed: 2026-09-05 · Sources cited below.